Nevirapine

Generic Name: Nevirapine

Brand Names:

Availability:

Drug Class: non-nucleoside reverse transcriptase inhibitors (NNRTIs)

Therapeutic action

  • Antiretroviral, HIV-1 non nucleoside reverse transcriptase inhibitor

Indications

  • HIV-1 infection in neonates,in combination with other antiretrovirals

Forms and strengths

  • 50 mg/5 ml oral suspension

Dosage

The daily dose is administered in 2 divided doses.

  • Child under one month:

 

Weight

50 mg/5 ml oral suspension (10 mg/ml)
2 to < 3 kg1.5 ml x 2
3 to < 4 kg2 ml x 2
4 to < 5 kg3 ml x 2

Duration

Change to lopinavir/ritonavir granules(at 2 weeks of age) or dolutegravir dispersible tablet (at 4 weeks of age).

Contra-indications, adverse effects, precautions

  • May cause:
  • cutaneous reactions sometimes severe (Stevens-Johnson and Lyell syndromes), hepatic disorders possibly severe (fulminant hepatitis) and haematological disorders. In these cases, stop nevirapine immediately and permanently;
  • gastrointestinal disturbances (take with food to increase tolerance), headache, myalgia.
  • Avoid combination with rifampicin (decreases the efficacy of nevirapine).

Remarks

  • Nevirapine is also used for prophylactic treatment to reduce mother-to-child transmission and treatment of HIV-1 infection in children and adults, in combination with other antiretrovirals. Check national recommendations.

Storage

Below 25 °C

Once opened, oral suspension keeps for 2 months maximum.